Lack of selectivity of URB602 for 2-oleoylglycerol compared to anandamide hydrolysis in vitro.
Vandevoorde, S
Lack of selectivity of URB602 for 2-oleoylglycerol compared to anandamide hydrolysis in vitro. [electronic resource] - British journal of pharmacology Jan 2007 - 186-91 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
0007-1188
10.1038/sj.bjp.0706971 doi
Amidohydrolases--antagonists & inhibitors
Aniline Compounds--pharmacology
Animals
Arachidonic Acids--metabolism
Benzoxazines--pharmacology
Biphenyl Compounds--pharmacology
Cell Line, Tumor
Cells, Cultured
Cerebellum--metabolism
Cytosol--metabolism
Endocannabinoids
Glycerides--metabolism
Humans
Hydrolysis
In Vitro Techniques
Male
Membranes--metabolism
Mice
Monoacylglycerol Lipases--antagonists & inhibitors
Polyunsaturated Alkamides--metabolism
Rats
Rats, Wistar
Recombinant Proteins--antagonists & inhibitors
Lack of selectivity of URB602 for 2-oleoylglycerol compared to anandamide hydrolysis in vitro. [electronic resource] - British journal of pharmacology Jan 2007 - 186-91 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
0007-1188
10.1038/sj.bjp.0706971 doi
Amidohydrolases--antagonists & inhibitors
Aniline Compounds--pharmacology
Animals
Arachidonic Acids--metabolism
Benzoxazines--pharmacology
Biphenyl Compounds--pharmacology
Cell Line, Tumor
Cells, Cultured
Cerebellum--metabolism
Cytosol--metabolism
Endocannabinoids
Glycerides--metabolism
Humans
Hydrolysis
In Vitro Techniques
Male
Membranes--metabolism
Mice
Monoacylglycerol Lipases--antagonists & inhibitors
Polyunsaturated Alkamides--metabolism
Rats
Rats, Wistar
Recombinant Proteins--antagonists & inhibitors