Comparative effects of some hydrophilic excipients on the rate of gabapentin and baclofen lactamization in lyophilized formulations.

Cutrignelli, Annalisa

Comparative effects of some hydrophilic excipients on the rate of gabapentin and baclofen lactamization in lyophilized formulations. [electronic resource] - International journal of pharmaceutics Mar 2007 - 98-106 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

0378-5173

10.1016/j.ijpharm.2006.09.053 doi


Amines--chemistry
Anticonvulsants--chemistry
Baclofen--chemistry
Calorimetry, Differential Scanning
Chemistry, Pharmaceutical
Cyclohexanecarboxylic Acids--chemistry
Drug Stability
Excipients--chemistry
Freeze Drying
Gabapentin
Humidity
Kinetics
Lactams--chemistry
Lactose--chemistry
Mannitol--chemistry
Models, Chemical
Molecular Structure
Parasympatholytics--chemistry
Povidone--chemistry
Raffinose--chemistry
Technology, Pharmaceutical--methods
Temperature
Thermogravimetry
Trehalose--chemistry
Water--chemistry
beta-Cyclodextrins--chemistry
gamma-Aminobutyric Acid--chemistry