In vivo evidence that 5-HT(2C) receptors inhibit 5-HT neuronal activity via a GABAergic mechanism.

Boothman, L

In vivo evidence that 5-HT(2C) receptors inhibit 5-HT neuronal activity via a GABAergic mechanism. [electronic resource] - British journal of pharmacology Dec 2006 - 861-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0007-1188

10.1038/sj.bjp.0706935 doi


Action Potentials--drug effects
Aminopyridines--pharmacology
Animals
Brain Chemistry--drug effects
Dopamine Agonists--metabolism
Dopamine Antagonists--pharmacology
Dose-Response Relationship, Drug
GABA Antagonists--pharmacology
Glutamate Decarboxylase--analysis
Immunohistochemistry
Indoles--pharmacology
Male
Neural Inhibition--drug effects
Neurons--chemistry
Picrotoxin--pharmacology
Piperazines--pharmacology
Positron-Emission Tomography
Proto-Oncogene Proteins c-fos--analysis
Pyrazines--metabolism
Pyridines--pharmacology
Quinoxalines--metabolism
Raphe Nuclei--chemistry
Rats
Rats, Sprague-Dawley
Receptor, Serotonin, 5-HT2C--analysis
Ritanserin--pharmacology
Serotonin--metabolism
gamma-Aminobutyric Acid--metabolism