Engineering of cytochrome P450 3A4 for enhanced peroxide-mediated substrate oxidation using directed evolution and site-directed mutagenesis.
Kumar, Santosh
Engineering of cytochrome P450 3A4 for enhanced peroxide-mediated substrate oxidation using directed evolution and site-directed mutagenesis. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Dec 2006 - 1958-65 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
0090-9556
10.1124/dmd.106.012054 doi
Benzene Derivatives--chemistry
Coumarins--metabolism
Cytochrome P-450 CYP3A--genetics
Directed Molecular Evolution
Hydrogen Peroxide--chemistry
Mutagenesis, Site-Directed
Oxidation-Reduction
Quinolines--metabolism
Testosterone--metabolism
Engineering of cytochrome P450 3A4 for enhanced peroxide-mediated substrate oxidation using directed evolution and site-directed mutagenesis. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Dec 2006 - 1958-65 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
0090-9556
10.1124/dmd.106.012054 doi
Benzene Derivatives--chemistry
Coumarins--metabolism
Cytochrome P-450 CYP3A--genetics
Directed Molecular Evolution
Hydrogen Peroxide--chemistry
Mutagenesis, Site-Directed
Oxidation-Reduction
Quinolines--metabolism
Testosterone--metabolism