Induction of G2/M phase arrest and apoptosis of human leukemia cells by potent antitumor triazoloacridinone C-1305.

Augustin, Ewa

Induction of G2/M phase arrest and apoptosis of human leukemia cells by potent antitumor triazoloacridinone C-1305. [electronic resource] - Biochemical pharmacology Dec 2006 - 1668-79 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0006-2952

10.1016/j.bcp.2006.07.035 doi


Acridines--chemistry
Adenosine Triphosphate--metabolism
Antineoplastic Agents--chemistry
Apoptosis--drug effects
Blotting, Western
Caspase 3--metabolism
Cell Division--drug effects
Cell Line, Tumor
Cell Proliferation--drug effects
Electrophoresis, Agar Gel
Flow Cytometry
G2 Phase--drug effects
HL-60 Cells
Humans
In Situ Nick-End Labeling
Intracellular Membranes--drug effects
Leukemia
Membrane Potentials--drug effects
Mitochondria--drug effects
Poly (ADP-Ribose) Polymerase-1
Poly(ADP-ribose) Polymerases--metabolism
Triazoles--chemistry