Identification of isothiazole-4-carboxamidines derivatives as a novel class of allosteric MEK1 inhibitors.
El Abdellaoui, Hassan
Identification of isothiazole-4-carboxamidines derivatives as a novel class of allosteric MEK1 inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Nov 2006 - 5561-6 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2006.08.048 doi
Allosteric Regulation
Amidines--chemical synthesis
Animals
MAP Kinase Kinase 1--antagonists & inhibitors
MAP Kinase Kinase 2--antagonists & inhibitors
Rats
Identification of isothiazole-4-carboxamidines derivatives as a novel class of allosteric MEK1 inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters Nov 2006 - 5561-6 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2006.08.048 doi
Allosteric Regulation
Amidines--chemical synthesis
Animals
MAP Kinase Kinase 1--antagonists & inhibitors
MAP Kinase Kinase 2--antagonists & inhibitors
Rats