A medicinal-chemistry-guided approach to selective and druglike sigma 1 ligands.

Corbera, Jordi

A medicinal-chemistry-guided approach to selective and druglike sigma 1 ligands. [electronic resource] - ChemMedChem Jan 2006 - 140-54 p. digital

Publication Type: Journal Article

1860-7179

10.1002/cmdc.200500034 doi


Animals
Caco-2 Cells
Humans
Ligands
Magnetic Resonance Spectroscopy
Mass Spectrometry
Microsomes, Liver--metabolism
Protein Binding
Rats
Receptors, sigma--metabolism
Structure-Activity Relationship