In vitro and in vivo characterization of F-97013-GD, a partial 5-HT1A agonist with antipsychotic- and antiparkinsonian-like properties.

Zazpe, Arturo

In vitro and in vivo characterization of F-97013-GD, a partial 5-HT1A agonist with antipsychotic- and antiparkinsonian-like properties. [electronic resource] - Neuropharmacology Jul 2006 - 129-40 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0028-3908

10.1016/j.neuropharm.2006.03.008 doi


5-Hydroxytryptophan--pharmacology
Animals
Antiparkinson Agents--pharmacology
Antipsychotic Agents--pharmacology
Apomorphine--pharmacology
Avoidance Learning--drug effects
Binding, Competitive--drug effects
Catalepsy--chemically induced
Dopamine Agonists--pharmacology
Dopamine D2 Receptor Antagonists
Dopamine Plasma Membrane Transport Proteins--metabolism
Drug Interactions
Guanosine 5'-O-(3-Thiotriphosphate)--metabolism
Haloperidol--antagonists & inhibitors
Head Movements--drug effects
Hypothermia--chemically induced
Jaw--physiology
Male
Mice
Motor Activity--drug effects
Piperazines--metabolism
Pyridazines--pharmacology
Pyridines--metabolism
Rats
Rats, Wistar
Receptor, Serotonin, 5-HT1A--drug effects
Receptors, Dopamine D2--metabolism
Serotonin Antagonists--metabolism
Serotonin Receptor Agonists--pharmacology
Tremor--physiopathology