Binding characteristics of levetiracetam to synaptic vesicle protein 2A (SV2A) in human brain and in CHO cells expressing the human recombinant protein.

Gillard, Michel

Binding characteristics of levetiracetam to synaptic vesicle protein 2A (SV2A) in human brain and in CHO cells expressing the human recombinant protein. [electronic resource] - European journal of pharmacology Apr 2006 - 102-8 p. digital

Publication Type: Journal Article

0014-2999

10.1016/j.ejphar.2006.02.022 doi


Animals
Azides--metabolism
Binding Sites
Binding, Competitive
Brain--metabolism
CHO Cells
Cerebellum--metabolism
Cerebral Cortex--metabolism
Cricetinae
Cricetulus
Female
Gene Expression
Hippocampus--metabolism
Humans
Kinetics
Levetiracetam
Male
Membrane Glycoproteins--genetics
Nerve Tissue Proteins--genetics
Piracetam--analogs & derivatives
Pyrrolidines--metabolism
Recombinant Proteins--metabolism
Tritium