Synthesis and SAR of highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drugs.

Kling, Andreas

Synthesis and SAR of highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drugs. [electronic resource] - Bioorganic & medicinal chemistry letters Dec 2005 - 5567-73 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2005.04.077 doi


Antidepressive Agents--chemical synthesis
Humans
Indoles--chemistry
Kinetics
Models, Molecular
Piperazines--chemistry
Serotonin 5-HT1 Receptor Antagonists
Structure-Activity Relationship