Intrinsic efficacy of antipsychotics at human D2, D3, and D4 dopamine receptors: identification of the clozapine metabolite N-desmethylclozapine as a D2/D3 partial agonist.

Burstein, E S

Intrinsic efficacy of antipsychotics at human D2, D3, and D4 dopamine receptors: identification of the clozapine metabolite N-desmethylclozapine as a D2/D3 partial agonist. [electronic resource] - The Journal of pharmacology and experimental therapeutics Dec 2005 - 1278-87 p. digital

Publication Type: Comparative Study; Journal Article

0022-3565

10.1124/jpet.105.092155 doi


Animals
Antipsychotic Agents--metabolism
Clozapine--metabolism
Haloperidol--pharmacology
Humans
Mice
NIH 3T3 Cells
Pergolide--pharmacology
Plasmids
RGS Proteins--metabolism
Receptors, Dopamine D2--agonists
Receptors, Dopamine D3--agonists
Receptors, Dopamine D4--metabolism
Transfection