Electrophysiological and in vivo characterization of A-317567, a novel blocker of acid sensing ion channels.

Dubé, G R

Electrophysiological and in vivo characterization of A-317567, a novel blocker of acid sensing ion channels. [electronic resource] - Pain Sep 2005 - 88-96 p. digital

Publication Type: Comparative Study; Journal Article

0304-3959

10.1016/j.pain.2005.05.021 doi


Acid Sensing Ion Channels
Acids--pharmacology
Amiloride--analogs & derivatives
Animals
Cell Count--methods
Cell Size
Disease Models, Animal
Dose-Response Relationship, Drug
Drug Interactions
Freund's Adjuvant
Ganglia, Spinal--cytology
Hydrogen-Ion Concentration
Hyperalgesia--chemically induced
Isoquinolines--pharmacology
Membrane Potentials--drug effects
Membrane Proteins--classification
Naphthalenes--pharmacology
Nerve Tissue Proteins--classification
Neurons--drug effects
Pain Measurement--methods
Pain Threshold--drug effects
Pain, Postoperative--chemically induced
Patch-Clamp Techniques--methods
Rats
Rats, Sprague-Dawley
Sodium Channels--classification