A fluoroquinolone resistance protein from Mycobacterium tuberculosis that mimics DNA.
Hegde, Subray S
A fluoroquinolone resistance protein from Mycobacterium tuberculosis that mimics DNA. [electronic resource] - Science (New York, N.Y.) Jun 2005 - 1480-3 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
1095-9203
10.1126/science.1110699 doi
Amino Acid Sequence
Antitubercular Agents--chemistry
Bacterial Proteins--chemistry
Ciprofloxacin--pharmacology
Crystallography, X-Ray
DNA Gyrase--metabolism
DNA, Bacterial--chemistry
DNA, Superhelical--chemistry
Drug Resistance, Bacterial
Drug Resistance, Microbial--physiology
Enzyme Inhibitors--chemistry
Escherichia coli--enzymology
Fluoroquinolones--antagonists & inhibitors
Models, Molecular
Molecular Mimicry
Molecular Sequence Data
Monomeric GTP-Binding Proteins
Mycobacterium tuberculosis--drug effects
Protein Conformation
Protein Folding
Structure-Activity Relationship
Topoisomerase II Inhibitors
A fluoroquinolone resistance protein from Mycobacterium tuberculosis that mimics DNA. [electronic resource] - Science (New York, N.Y.) Jun 2005 - 1480-3 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
1095-9203
10.1126/science.1110699 doi
Amino Acid Sequence
Antitubercular Agents--chemistry
Bacterial Proteins--chemistry
Ciprofloxacin--pharmacology
Crystallography, X-Ray
DNA Gyrase--metabolism
DNA, Bacterial--chemistry
DNA, Superhelical--chemistry
Drug Resistance, Bacterial
Drug Resistance, Microbial--physiology
Enzyme Inhibitors--chemistry
Escherichia coli--enzymology
Fluoroquinolones--antagonists & inhibitors
Models, Molecular
Molecular Mimicry
Molecular Sequence Data
Monomeric GTP-Binding Proteins
Mycobacterium tuberculosis--drug effects
Protein Conformation
Protein Folding
Structure-Activity Relationship
Topoisomerase II Inhibitors