Neuropharmacokinetics of a new alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid (AMPA) modulator, S18986 [(S)-2,3-dihydro-[3,4]cyclopentano-1,2,4-benzothiadiazine-1,1-dioxide], in the rat.

Bourasset, Fanchon

Neuropharmacokinetics of a new alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid (AMPA) modulator, S18986 [(S)-2,3-dihydro-[3,4]cyclopentano-1,2,4-benzothiadiazine-1,1-dioxide], in the rat. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Aug 2005 - 1137-43 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0090-9556

10.1124/dmd.105.004424 doi


Allosteric Regulation
Animals
Benzothiadiazines--administration & dosage
Blood-Brain Barrier--metabolism
Brain--metabolism
Brain Chemistry
Extracellular Fluid--metabolism
Frontal Lobe--metabolism
Hippocampus--metabolism
Intracellular Fluid--metabolism
Male
Microdialysis
Molecular Structure
Perfusion
Rats
Rats, Wistar
Receptors, AMPA--metabolism