The effects of subunit composition on the inhibition of nicotinic receptors by the amphipathic blocker 2,2,6,6-tetramethylpiperidin-4-yl heptanoate.
Papke, Roger L
The effects of subunit composition on the inhibition of nicotinic receptors by the amphipathic blocker 2,2,6,6-tetramethylpiperidin-4-yl heptanoate. [electronic resource] - Molecular pharmacology Jun 2005 - 1977-90 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
0026-895X
10.1124/mol.105.011676 doi
Amino Acid Sequence
Animals
Dose-Response Relationship, Drug
Female
Heptanoic Acids--chemistry
Male
Mice
Molecular Sequence Data
Nicotinic Antagonists--chemistry
Piperidines--chemistry
Protein Subunits--antagonists & inhibitors
Rats
Rats, Sprague-Dawley
Receptors, Nicotinic--chemistry
Xenopus laevis
The effects of subunit composition on the inhibition of nicotinic receptors by the amphipathic blocker 2,2,6,6-tetramethylpiperidin-4-yl heptanoate. [electronic resource] - Molecular pharmacology Jun 2005 - 1977-90 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
0026-895X
10.1124/mol.105.011676 doi
Amino Acid Sequence
Animals
Dose-Response Relationship, Drug
Female
Heptanoic Acids--chemistry
Male
Mice
Molecular Sequence Data
Nicotinic Antagonists--chemistry
Piperidines--chemistry
Protein Subunits--antagonists & inhibitors
Rats
Rats, Sprague-Dawley
Receptors, Nicotinic--chemistry
Xenopus laevis