Do drug substrates enter the common drug-binding pocket of P-glycoprotein through "gates"?
Loo, Tip W
Do drug substrates enter the common drug-binding pocket of P-glycoprotein through "gates"? [electronic resource] - Biochemical and biophysical research communications Apr 2005 - 419-22 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0006-291X
10.1016/j.bbrc.2005.01.134 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--chemistry
Animals
Binding Sites
Drug Resistance--physiology
Humans
Ion Channel Gating--physiology
Models, Biological
Models, Chemical
Pharmaceutical Preparations--chemistry
Protein Binding
Protein Conformation
Structure-Activity Relationship
Do drug substrates enter the common drug-binding pocket of P-glycoprotein through "gates"? [electronic resource] - Biochemical and biophysical research communications Apr 2005 - 419-22 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0006-291X
10.1016/j.bbrc.2005.01.134 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--chemistry
Animals
Binding Sites
Drug Resistance--physiology
Humans
Ion Channel Gating--physiology
Models, Biological
Models, Chemical
Pharmaceutical Preparations--chemistry
Protein Binding
Protein Conformation
Structure-Activity Relationship