Extravascular transport of drugs in tumor tissue: effect of lipophilicity on diffusion of tirapazamine analogues in multicellular layer cultures.

Pruijn, Frederik B

Extravascular transport of drugs in tumor tissue: effect of lipophilicity on diffusion of tirapazamine analogues in multicellular layer cultures. [electronic resource] - Journal of medicinal chemistry Feb 2005 - 1079-87 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0022-2623

10.1021/jm049549p doi


Antineoplastic Agents--chemistry
Biological Transport
Diffusion
HT29 Cells
Humans
Models, Biological
Solubility
Tirapazamine
Triazines--chemistry