Synthesis and SAR of 5,6-diarylpyridines as human CB1 inverse agonists.
Meurer, Laura C
Synthesis and SAR of 5,6-diarylpyridines as human CB1 inverse agonists. [electronic resource] - Bioorganic & medicinal chemistry letters Feb 2005 - 645-51 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2004.11.031 doi
Animals
Biological Availability
CHO Cells
Cricetinae
Humans
Inhibitory Concentration 50
Male
Pyridines--chemical synthesis
Radioligand Assay
Rats
Rats, Sprague-Dawley
Receptor, Cannabinoid, CB1--agonists
Structure-Activity Relationship
Tissue Distribution
Transfection
Synthesis and SAR of 5,6-diarylpyridines as human CB1 inverse agonists. [electronic resource] - Bioorganic & medicinal chemistry letters Feb 2005 - 645-51 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2004.11.031 doi
Animals
Biological Availability
CHO Cells
Cricetinae
Humans
Inhibitory Concentration 50
Male
Pyridines--chemical synthesis
Radioligand Assay
Rats
Rats, Sprague-Dawley
Receptor, Cannabinoid, CB1--agonists
Structure-Activity Relationship
Tissue Distribution
Transfection