The novel estrogen 17alpha-20Z-21-[(4-amino)phenyl]-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diol induces apoptosis in prostate cancer cell lines at nanomolar concentrations in vitro.

Mobley, James A

The novel estrogen 17alpha-20Z-21-[(4-amino)phenyl]-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diol induces apoptosis in prostate cancer cell lines at nanomolar concentrations in vitro. [electronic resource] - Molecular cancer therapeutics May 2004 - 587-95 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.; Research Support, U.S. Gov't, P.H.S.

1535-7163


Apoptosis--drug effects
Blotting, Western
Bromodeoxyuridine
Caspase 3
Caspases--metabolism
Cell Cycle--drug effects
Cell Line, Tumor
Drug Screening Assays, Antitumor
Estradiol--analogs & derivatives
Estrogen Receptor alpha--metabolism
Estrogen Receptor beta--metabolism
Flow Cytometry
Humans
Male
Models, Molecular
Prostatic Neoplasms--pathology
Protein Binding