Ritonavir and dexamethasone induce expression of CYP3A and P-glycoprotein in rats.
Perloff, M D
Ritonavir and dexamethasone induce expression of CYP3A and P-glycoprotein in rats. [electronic resource] - Xenobiotica; the fate of foreign compounds in biological systems Feb 2004 - 133-50 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
0049-8254
10.1080/00498250310001630215 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--biosynthesis
Algorithms
Animals
Anti-Inflammatory Agents--pharmacology
Antibodies, Blocking--pharmacology
Aryl Hydrocarbon Hydroxylases--antagonists & inhibitors
Blood-Brain Barrier--drug effects
Blotting, Western
Capillaries--drug effects
Chromatography, High Pressure Liquid
Cytochrome P-450 CYP3A
Dexamethasone--pharmacology
Enzyme Induction--drug effects
Enzyme Inhibitors--pharmacology
GABA Modulators--metabolism
Gene Expression--drug effects
HIV Protease Inhibitors--pharmacology
Intestines--drug effects
Liver--drug effects
Luminescent Measurements
Male
Microsomes--drug effects
Oxidoreductases, N-Demethylating--antagonists & inhibitors
Rats
Rats, Sprague-Dawley
Ritonavir--pharmacology
Triazolam--metabolism
Ritonavir and dexamethasone induce expression of CYP3A and P-glycoprotein in rats. [electronic resource] - Xenobiotica; the fate of foreign compounds in biological systems Feb 2004 - 133-50 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
0049-8254
10.1080/00498250310001630215 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--biosynthesis
Algorithms
Animals
Anti-Inflammatory Agents--pharmacology
Antibodies, Blocking--pharmacology
Aryl Hydrocarbon Hydroxylases--antagonists & inhibitors
Blood-Brain Barrier--drug effects
Blotting, Western
Capillaries--drug effects
Chromatography, High Pressure Liquid
Cytochrome P-450 CYP3A
Dexamethasone--pharmacology
Enzyme Induction--drug effects
Enzyme Inhibitors--pharmacology
GABA Modulators--metabolism
Gene Expression--drug effects
HIV Protease Inhibitors--pharmacology
Intestines--drug effects
Liver--drug effects
Luminescent Measurements
Male
Microsomes--drug effects
Oxidoreductases, N-Demethylating--antagonists & inhibitors
Rats
Rats, Sprague-Dawley
Ritonavir--pharmacology
Triazolam--metabolism