Muscarinic M2 receptor stimulation of Cav1.2b requires phosphatidylinositol 3-kinase, protein kinase C, and c-Src.
Callaghan, B
Muscarinic M2 receptor stimulation of Cav1.2b requires phosphatidylinositol 3-kinase, protein kinase C, and c-Src. [electronic resource] - Circulation research Mar 2004 - 626-33 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
1524-4571
10.1161/01.RES.0000118248.17466.B7 doi
Acetylcholine--pharmacology
Animals
Barium--metabolism
Calcium Channels, L-Type--physiology
Carbazoles--pharmacology
Cells, Cultured--drug effects
Chromones--pharmacology
Class Ib Phosphatidylinositol 3-Kinase
Diamines--pharmacology
Enzyme Inhibitors--pharmacology
GTP-Binding Protein beta Subunits--antagonists & inhibitors
GTP-Binding Protein gamma Subunits--antagonists & inhibitors
Indoles--pharmacology
Ion Channel Gating--drug effects
Ion Transport--drug effects
Isoenzymes--antagonists & inhibitors
Male
Morpholines--pharmacology
Muscarinic Agonists--pharmacology
Muscarinic Antagonists--pharmacology
Muscle, Smooth, Vascular--cytology
Myocytes, Smooth Muscle--drug effects
Naphthalenes--pharmacology
Patch-Clamp Techniques
Phorbol 12,13-Dibutyrate--pharmacology
Phosphatidylinositol 3-Kinases--physiology
Phosphoinositide-3 Kinase Inhibitors
Piperidines--pharmacology
Portal Vein--cytology
Protein Kinase C--antagonists & inhibitors
Proto-Oncogene Proteins pp60(c-src)--antagonists & inhibitors
Pyrimidines--pharmacology
Rabbits
Receptor, Muscarinic M2--agonists
Receptor, Muscarinic M3--drug effects
Signal Transduction--drug effects
Muscarinic M2 receptor stimulation of Cav1.2b requires phosphatidylinositol 3-kinase, protein kinase C, and c-Src. [electronic resource] - Circulation research Mar 2004 - 626-33 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
1524-4571
10.1161/01.RES.0000118248.17466.B7 doi
Acetylcholine--pharmacology
Animals
Barium--metabolism
Calcium Channels, L-Type--physiology
Carbazoles--pharmacology
Cells, Cultured--drug effects
Chromones--pharmacology
Class Ib Phosphatidylinositol 3-Kinase
Diamines--pharmacology
Enzyme Inhibitors--pharmacology
GTP-Binding Protein beta Subunits--antagonists & inhibitors
GTP-Binding Protein gamma Subunits--antagonists & inhibitors
Indoles--pharmacology
Ion Channel Gating--drug effects
Ion Transport--drug effects
Isoenzymes--antagonists & inhibitors
Male
Morpholines--pharmacology
Muscarinic Agonists--pharmacology
Muscarinic Antagonists--pharmacology
Muscle, Smooth, Vascular--cytology
Myocytes, Smooth Muscle--drug effects
Naphthalenes--pharmacology
Patch-Clamp Techniques
Phorbol 12,13-Dibutyrate--pharmacology
Phosphatidylinositol 3-Kinases--physiology
Phosphoinositide-3 Kinase Inhibitors
Piperidines--pharmacology
Portal Vein--cytology
Protein Kinase C--antagonists & inhibitors
Proto-Oncogene Proteins pp60(c-src)--antagonists & inhibitors
Pyrimidines--pharmacology
Rabbits
Receptor, Muscarinic M2--agonists
Receptor, Muscarinic M3--drug effects
Signal Transduction--drug effects