Design and synthesis of aminopropyl tetrahydroindole-based indolin-2-ones as selective and potent inhibitors of Src and Yes tyrosine kinase.

Guan, Huiping

Design and synthesis of aminopropyl tetrahydroindole-based indolin-2-ones as selective and potent inhibitors of Src and Yes tyrosine kinase. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2004 - 187-90 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2003.09.069 doi


Drug Design
Enzyme Inhibitors--chemical synthesis
Indoles--chemical synthesis
Structure-Activity Relationship
src-Family Kinases--antagonists & inhibitors