The influence of the P-glycoprotein inhibitor zosuquidar trihydrochloride (LY335979) on the brain penetration of paclitaxel in mice.
Kemper, E Marleen
The influence of the P-glycoprotein inhibitor zosuquidar trihydrochloride (LY335979) on the brain penetration of paclitaxel in mice. [electronic resource] - Cancer chemotherapy and pharmacology Feb 2004 - 173-8 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0344-5704
10.1007/s00280-003-0720-y doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Administration, Oral
Algorithms
Animals
Antineoplastic Agents, Phytogenic--pharmacokinetics
Area Under Curve
Biological Availability
Brain--drug effects
Dibenzocycloheptenes--pharmacology
Female
Injections, Intravenous
Mice
Mice, Knockout
Paclitaxel--pharmacokinetics
Quinolines--pharmacology
Spectrophotometry, Ultraviolet
Tissue Distribution
The influence of the P-glycoprotein inhibitor zosuquidar trihydrochloride (LY335979) on the brain penetration of paclitaxel in mice. [electronic resource] - Cancer chemotherapy and pharmacology Feb 2004 - 173-8 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0344-5704
10.1007/s00280-003-0720-y doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Administration, Oral
Algorithms
Animals
Antineoplastic Agents, Phytogenic--pharmacokinetics
Area Under Curve
Biological Availability
Brain--drug effects
Dibenzocycloheptenes--pharmacology
Female
Injections, Intravenous
Mice
Mice, Knockout
Paclitaxel--pharmacokinetics
Quinolines--pharmacology
Spectrophotometry, Ultraviolet
Tissue Distribution