Lack of intrinsic activity and significant subtype selectivity of SR 95639A at muscarinic receptors.

Mohamed, A S

Lack of intrinsic activity and significant subtype selectivity of SR 95639A at muscarinic receptors. [electronic resource] - European journal of pharmacology Oct 1992 - 181-7 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.; Research Support, U.S. Gov't, P.H.S.

0014-2999

10.1016/0922-4106(92)90126-g doi


Acetylcholine--metabolism
Animals
Binding Sites
CHO Cells
Carbachol--pharmacology
Cerebral Cortex--drug effects
Colforsin--pharmacology
Cricetinae
Cyclic AMP--metabolism
Female
Hydrolysis
Inositol Phosphates--metabolism
Male
Morpholines--metabolism
N-Methylscopolamine
Pyridazines--metabolism
Rats
Rats, Sprague-Dawley
Receptors, Muscarinic--drug effects
Scopolamine Derivatives--metabolism
Transfection