Comparison of the functional blockade of rat substance P (NK1) receptors by GR205171, RP67580, SR140333 and NKP-608.

Rupniak, Nadia M J

Comparison of the functional blockade of rat substance P (NK1) receptors by GR205171, RP67580, SR140333 and NKP-608. [electronic resource] - Neuropharmacology Aug 2003 - 231-41 p. digital

Publication Type: Comparative Study; Journal Article

0028-3908

10.1016/s0028-3908(03)00157-6 doi


Animals
CHO Cells
Cricetinae
Dose-Response Relationship, Drug
Female
Gerbillinae
Humans
Indoles--metabolism
Isoindoles
Male
Neurokinin-1 Receptor Antagonists
Piperidines--metabolism
Quinolines--metabolism
Quinuclidines--metabolism
Rats
Rats, Sprague-Dawley
Receptors, Neurokinin-1--metabolism
Tetrazoles--metabolism
Tumor Cells, Cultured