Receptor occupancy of nonpeptide corticotropin-releasing factor 1 antagonist DMP696: correlation with drug exposure and anxiolytic efficacy.

Li, Yu-Wen

Receptor occupancy of nonpeptide corticotropin-releasing factor 1 antagonist DMP696: correlation with drug exposure and anxiolytic efficacy. [electronic resource] - The Journal of pharmacology and experimental therapeutics Apr 2003 - 86-96 p. digital

Publication Type: Journal Article

0022-3565

10.1124/jpet.102.045914 doi


Amphibian Proteins
Animals
Anxiety--blood
Binding Sites
Corticotropin-Releasing Hormone--metabolism
Disease Models, Animal
Drug Interactions
Iodine Radioisotopes
Male
Peptide Hormones
Peptides--metabolism
Pyrazoles--blood
Rats
Rats, Sprague-Dawley
Receptors, Corticotropin-Releasing Hormone--antagonists & inhibitors
Statistics as Topic
Substance Withdrawal Syndrome
Time Factors
Triazines--blood
CRF Receptor, Type 1