Role of human MDR1 gene polymorphism in bioavailability and interaction of digoxin, a substrate of P-glycoprotein.
Kurata, Yasuo
Role of human MDR1 gene polymorphism in bioavailability and interaction of digoxin, a substrate of P-glycoprotein. [electronic resource] - Clinical pharmacology and therapeutics Aug 2002 - 209-19 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0009-9236
10.1067/mcp.2002.126177 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
Administration, Oral
Adult
Alleles
Anti-Bacterial Agents--pharmacokinetics
Area Under Curve
Asian People--genetics
Biological Availability
Cardiotonic Agents--pharmacokinetics
Clarithromycin--administration & dosage
Cytochrome P-450 Enzyme System--metabolism
Digoxin--administration & dosage
Drug Administration Schedule
Drug Interactions
Enzyme Inhibitors--pharmacokinetics
Genes, MDR
Genotype
Humans
Injections, Intravenous
Japan
Male
Polymerase Chain Reaction
Polymorphism, Genetic
Polymorphism, Restriction Fragment Length
Reference Values
Role of human MDR1 gene polymorphism in bioavailability and interaction of digoxin, a substrate of P-glycoprotein. [electronic resource] - Clinical pharmacology and therapeutics Aug 2002 - 209-19 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0009-9236
10.1067/mcp.2002.126177 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
Administration, Oral
Adult
Alleles
Anti-Bacterial Agents--pharmacokinetics
Area Under Curve
Asian People--genetics
Biological Availability
Cardiotonic Agents--pharmacokinetics
Clarithromycin--administration & dosage
Cytochrome P-450 Enzyme System--metabolism
Digoxin--administration & dosage
Drug Administration Schedule
Drug Interactions
Enzyme Inhibitors--pharmacokinetics
Genes, MDR
Genotype
Humans
Injections, Intravenous
Japan
Male
Polymerase Chain Reaction
Polymorphism, Genetic
Polymorphism, Restriction Fragment Length
Reference Values