Synthesis and structure-activity relationships of M(2)-selective muscarinic receptor ligands in the 1-[4-(4-arylsulfonyl)-phenylmethyl]-4-(4-piperidinyl)-piperazine family.

McCombie, Stuart W

Synthesis and structure-activity relationships of M(2)-selective muscarinic receptor ligands in the 1-[4-(4-arylsulfonyl)-phenylmethyl]-4-(4-piperidinyl)-piperazine family. [electronic resource] - Bioorganic & medicinal chemistry letters Mar 2002 - 795-8 p. digital

Publication Type: Journal Article

0960-894X

10.1016/s0960-894x(02)00024-0 doi


Binding Sites
Ligands
Molecular Structure
Piperazines--chemical synthesis
Receptor, Muscarinic M1
Receptor, Muscarinic M2
Receptors, Muscarinic--metabolism
Structure-Activity Relationship