Evaluation of farnesyl:protein transferase and geranylgeranyl:protein transferase inhibitor combinations in preclinical models.

Lobell, R B

Evaluation of farnesyl:protein transferase and geranylgeranyl:protein transferase inhibitor combinations in preclinical models. [electronic resource] - Cancer research Dec 2001 - 8758-68 p. digital

Publication Type: Comparative Study; Evaluation Study; Journal Article

0008-5472


Alkyl and Aryl Transferases--antagonists & inhibitors
Animals
Antineoplastic Combined Chemotherapy Protocols--pharmacology
Apoptosis--drug effects
Drug Screening Assays, Antitumor
Drug Synergism
Enzyme Inhibitors--administration & dosage
Farnesyltranstransferase
Female
Humans
Mice
Mice, Nude
Pancreatic Neoplasms--drug therapy
Protein Prenylation--drug effects
Tumor Cells, Cultured
Xenograft Model Antitumor Assays
ras Proteins--metabolism