Analysis of binding domain and function of chimeric mu/kappa opioid receptors to ohmefentanyl stereoisomers.
Feng, Y P
Analysis of binding domain and function of chimeric mu/kappa opioid receptors to ohmefentanyl stereoisomers. [electronic resource] - Acta pharmacologica Sinica Nov 2001 - 981-5 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1671-4083
3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer--pharmacology
Analgesics--pharmacology
Animals
Binding Sites
COS Cells--metabolism
Chlorocebus aethiops
Cyclic AMP--metabolism
Dynorphins--metabolism
Fentanyl--analogs & derivatives
Peptide Fragments--metabolism
Protein Structure, Tertiary
Receptors, Opioid, kappa--metabolism
Receptors, Opioid, mu--metabolism
Recombinant Fusion Proteins--metabolism
Stereoisomerism
Analysis of binding domain and function of chimeric mu/kappa opioid receptors to ohmefentanyl stereoisomers. [electronic resource] - Acta pharmacologica Sinica Nov 2001 - 981-5 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1671-4083
3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer--pharmacology
Analgesics--pharmacology
Animals
Binding Sites
COS Cells--metabolism
Chlorocebus aethiops
Cyclic AMP--metabolism
Dynorphins--metabolism
Fentanyl--analogs & derivatives
Peptide Fragments--metabolism
Protein Structure, Tertiary
Receptors, Opioid, kappa--metabolism
Receptors, Opioid, mu--metabolism
Recombinant Fusion Proteins--metabolism
Stereoisomerism