Design, synthesis, and biological activity of methoctramine-related polyamines as putative G(i) protein activators.

Melchiorre, C

Design, synthesis, and biological activity of methoctramine-related polyamines as putative G(i) protein activators. [electronic resource] - Journal of medicinal chemistry Nov 2001 - 4035-8 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-2623

10.1021/jm0155594 doi


Animals
Atrial Function
CHO Cells
Cricetinae
Diamines--chemistry
Drug Design
Electric Stimulation
GTP-Binding Protein alpha Subunits, Gi-Go--metabolism
Guinea Pigs
Heart Atria--drug effects
Humans
In Vitro Techniques
Muscarinic Agonists--pharmacology
Polyamines--chemical synthesis
Rats
Receptors, Muscarinic--metabolism
Structure-Activity Relationship