Activation of inositol 1,4,5-trisphosphate receptor is essential for the opening of mouse TRP5 channels.

Kanki, H

Activation of inositol 1,4,5-trisphosphate receptor is essential for the opening of mouse TRP5 channels. [electronic resource] - Molecular pharmacology Nov 2001 - 989-98 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0026-895X

10.1124/mol.60.5.989 doi


Acetylcholine--metabolism
Adenosine--analogs & derivatives
Allosteric Regulation
Animals
Calcium--deficiency
Calcium Channel Agonists--pharmacology
Calcium Channels--drug effects
Cation Transport Proteins
Electrophysiology
Estrenes--pharmacology
GTP-Binding Protein alpha Subunits, Gq-G11
GTP-Binding Proteins--metabolism
Guanosine 5'-O-(3-Thiotriphosphate)--metabolism
Heterotrimeric GTP-Binding Proteins--antagonists & inhibitors
Inositol 1,4,5-Trisphosphate--metabolism
Inositol 1,4,5-Trisphosphate Receptors
Macrocyclic Compounds
Mice
Nuclear Proteins--antagonists & inhibitors
Oligodeoxyribonucleotides, Antisense--pharmacology
Oocytes--drug effects
Oxazoles--pharmacology
Peptides--chemical synthesis
Phosphodiesterase Inhibitors--pharmacology
Protein Serine-Threonine Kinases
Pyrrolidinones--pharmacology
Receptor, Muscarinic M1
Receptors, Cytoplasmic and Nuclear--antagonists & inhibitors
Receptors, Muscarinic--metabolism
TRPC Cation Channels
Type C Phospholipases--antagonists & inhibitors
Xenopus laevis