Contribution of P-glycoprotein to the enhancing effects of dimethyl-beta-cyclodextrin on oral bioavailability of tacrolimus.

Arima, H

Contribution of P-glycoprotein to the enhancing effects of dimethyl-beta-cyclodextrin on oral bioavailability of tacrolimus. [electronic resource] - The Journal of pharmacology and experimental therapeutics May 2001 - 547-55 p. digital

Publication Type: Journal Article

0022-3565


ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
Animals
Antineoplastic Agents, Phytogenic--pharmacology
Area Under Curve
Biological Availability
Blotting, Western
Caco-2 Cells
Cyclodextrins--pharmacology
Drug Resistance, Neoplasm
Flow Cytometry
Humans
Immunosuppressive Agents--pharmacokinetics
Intestinal Absorption--drug effects
Male
Rats
Rats, Wistar
Reverse Transcriptase Polymerase Chain Reaction
Silver Staining
Solubility
Tacrolimus--pharmacokinetics
Vinblastine--pharmacology
beta-Cyclodextrins