Influence of phenylalanine-481 substitutions on the catalytic activity of cytochrome P450 2D6.

Hayhurst, G P

Influence of phenylalanine-481 substitutions on the catalytic activity of cytochrome P450 2D6. [electronic resource] - The Biochemical journal Apr 2001 - 373-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0264-6021

10.1042/0264-6021:3550373 doi


Alkylation
Catalysis
Cytochrome P-450 CYP2D6--chemistry
Debrisoquin--pharmacokinetics
Dextromethorphan--pharmacokinetics
Kinetics
Metoprolol--pharmacokinetics
Mutagenesis, Site-Directed
Oxidation-Reduction
Phenylalanine--metabolism
Substrate Specificity