A rational approach to the design and synthesis of a new bradykinin B(1) receptor antagonist.

Bedos, P

A rational approach to the design and synthesis of a new bradykinin B(1) receptor antagonist. [electronic resource] - Journal of medicinal chemistry Jun 2000 - 2387-94 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm990962k doi


Animals
Bradykinin Receptor Antagonists
CHO Cells
Cricetinae
Drug Design
In Vitro Techniques
Magnetic Resonance Spectroscopy
Muscle Contraction--drug effects
Muscle, Smooth, Vascular--drug effects
Oligopeptides--chemical synthesis
Receptor, Bradykinin B1
Structure-Activity Relationship
Thiazepines--chemical synthesis
Transfection
Umbilical Veins--drug effects