The synthesis and vasopressin (AVP) antagonist activity of a novel series of N-aroyl-2,4,5,6-tetrahydropyrazolo[3,4-d]thieno[3,2-b]azepines.

Albright, J D

The synthesis and vasopressin (AVP) antagonist activity of a novel series of N-aroyl-2,4,5,6-tetrahydropyrazolo[3,4-d]thieno[3,2-b]azepines. [electronic resource] - Bioorganic & medicinal chemistry letters Apr 2000 - 695-8 p. digital

Publication Type: Journal Article

0960-894X

10.1016/s0960-894x(00)00084-6 doi


Animals
Arginine Vasopressin--antagonists & inhibitors
Azepines--chemical synthesis
Rats
Receptors, Vasopressin--metabolism
Structure-Activity Relationship