Ligand recognition of serine-cysteine amino acid exchanges in transmembrane domain 5 of alpha2-adrenergic receptors by UK 14,304.

Cockcroft, V

Ligand recognition of serine-cysteine amino acid exchanges in transmembrane domain 5 of alpha2-adrenergic receptors by UK 14,304. [electronic resource] - Journal of neurochemistry Apr 2000 - 1705-10 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-3042

10.1046/j.1471-4159.2000.0741705.x doi


Adrenergic alpha-Agonists--metabolism
Adrenergic alpha-Antagonists--pharmacology
Animals
Binding Sites--physiology
Binding, Competitive
Brimonidine Tartrate
CHO Cells
Chlorpromazine--metabolism
Cricetinae
Cysteine--metabolism
Dopamine Antagonists--metabolism
Humans
Idazoxan--analogs & derivatives
Ligands
Mice
Models, Molecular
Molecular Sequence Data
Oxymetazoline--metabolism
Protein Structure, Tertiary
Quinoxalines--metabolism
Radioligand Assay
Receptors, Adrenergic, alpha-2--chemistry
Sequence Homology, Amino Acid
Serine--metabolism
Transfection
Tritium
Yohimbine--metabolism