myo-inositol 1,4,6-trisphosphorothioate and myo-inositol 1,3, 6-trisphosphorothioate: partial agonists with very low intrinsic activity at the platelet myo-inositol 1,4,5-trisphosphate receptor.

Murphy, C T

myo-inositol 1,4,6-trisphosphorothioate and myo-inositol 1,3, 6-trisphosphorothioate: partial agonists with very low intrinsic activity at the platelet myo-inositol 1,4,5-trisphosphate receptor. [electronic resource] - Molecular pharmacology Mar 2000 - 595-601 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0026-895X

10.1124/mol.57.3.595 doi


Animals
Blood Platelets--drug effects
Calcium--metabolism
Calcium Channels--metabolism
Cell Membrane--drug effects
In Vitro Techniques
Inositol 1,4,5-Trisphosphate--analogs & derivatives
Inositol 1,4,5-Trisphosphate Receptors
Organothiophosphorus Compounds--pharmacology
Permeability
Rabbits
Rats
Receptors, Cytoplasmic and Nuclear--metabolism
Tritium