Chemical inhibitors of cyclin-dependent kinases: insights into design from X-ray crystallographic studies.

Noble, M E

Chemical inhibitors of cyclin-dependent kinases: insights into design from X-ray crystallographic studies. [electronic resource] - Pharmacology & therapeutics - 269-78 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Review

0163-7258

10.1016/s0163-7258(98)00051-5 doi


Adenosine Triphosphate--metabolism
Binding Sites
Crystallography, X-Ray
Cyclins--physiology
Drug Design
Drug Interactions
Enzyme Inhibitors--therapeutic use
Humans
Molecular Structure
Phosphotransferases--antagonists & inhibitors
Sensitivity and Specificity