Pharmacologic characterization of GSK-961081 (TD-5959), a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties. [electronic resource]
Producer: 20141125Description: 190-9 p. digitalISSN:- 1521-0103
- Adrenergic beta-2 Receptor Antagonists -- adverse effects
- Albuterol -- analogs & derivatives
- Animals
- Bronchodilator Agents -- adverse effects
- CHO Cells
- Carbamates -- adverse effects
- Cricetinae
- Cricetulus
- Cyclic AMP -- metabolism
- Drug Evaluation, Preclinical
- Guinea Pigs
- HEK293 Cells
- Humans
- Lung -- drug effects
- Muscarinic Antagonists -- adverse effects
- Muscle Relaxation
- Muscle, Smooth -- drug effects
- Protein Binding
- Quinolones -- adverse effects
- Receptors, Adrenergic, beta -- metabolism
- Receptors, Muscarinic -- metabolism
- Salmeterol Xinafoate
- Scopolamine Derivatives -- pharmacokinetics
- Tiotropium Bromide
- Tissue Distribution
- Trachea -- drug effects
No physical items for this record
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
There are no comments on this title.
Log in to your account to post a comment.