Synthesis and insight into the structure-activity relationships of chalcones as antimalarial agents. [electronic resource]
Producer: 20130417Description: 31-45 p. digitalISSN:- 1520-4804
- Animals
- Antimalarials -- chemical synthesis
- Benzopyrans -- chemical synthesis
- Catalytic Domain
- Chalcones -- chemical synthesis
- Chromans -- chemical synthesis
- Crotalaria -- chemistry
- Cysteine Endopeptidases -- chemistry
- Cysteine Proteinase Inhibitors -- chemical synthesis
- Malaria -- drug therapy
- Male
- Mice
- Molecular Docking Simulation
- Parasitic Sensitivity Tests
- Plasmodium falciparum -- drug effects
- Plasmodium yoelii
- Rats
- Rats, Sprague-Dawley
- Small Molecule Libraries
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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