"True" antiandrogens-selective non-ligand-binding pocket disruptors of androgen receptor-coactivator interactions: novel tools for prostate cancer. [electronic resource]
Producer: 20120525Description: 1635-44 p. digitalISSN:- 1520-4804
- Androgen Antagonists -- chemical synthesis
- Antineoplastic Agents -- chemical synthesis
- Cell Proliferation -- drug effects
- Cell Survival -- drug effects
- Databases, Factual
- Drug Screening Assays, Antitumor
- Estrogen Receptor alpha -- metabolism
- Estrogen Receptor beta -- metabolism
- Fluorescence Polarization
- Fluorescence Resonance Energy Transfer
- Humans
- Hydrazines -- chemical synthesis
- Male
- Models, Molecular
- Nuclear Receptor Coactivators -- metabolism
- Prostate-Specific Antigen -- metabolism
- Prostatic Neoplasms -- drug therapy
- Receptors, Androgen -- metabolism
- Receptors, Glucocorticoid -- metabolism
- Receptors, Progesterone -- antagonists & inhibitors
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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