Optimization of propafenone analogues as antimalarial leads. [electronic resource]
Producer: 20120207Description: 7477-85 p. digitalISSN:- 1520-4804
- Animals
- Antimalarials -- chemical synthesis
- Cell Line
- Drug Resistance
- Female
- Humans
- In Vitro Techniques
- Ion Channels -- antagonists & inhibitors
- Male
- Membranes, Artificial
- Mice
- Microsomes, Liver -- metabolism
- Parasitic Sensitivity Tests
- Permeability
- Plasmodium falciparum -- drug effects
- Propafenone -- analogs & derivatives
- Solubility
- Stereoisomerism
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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