Formation and anti-tumor activity of uncommon in vitro and in vivo metabolites of CPI-613, a novel anti-tumor compound that selectively alters tumor energy metabolism. [electronic resource]
Producer: 20111227Description: 163-82 p. digitalISSN:- 1874-0758
- Animals
- Antineoplastic Agents -- metabolism
- Caprylates -- metabolism
- Cell Line, Tumor
- Chromatography, Liquid
- Glucuronides -- metabolism
- Half-Life
- Humans
- Liver -- metabolism
- Mice
- Microsomes, Liver -- metabolism
- Neoplasms -- drug therapy
- Oxidation-Reduction
- Rats
- Rats, Sprague-Dawley
- Species Specificity
- Sulfides -- metabolism
- Sulfoxides -- metabolism
- Swine
- Swine, Miniature
- Tandem Mass Spectrometry
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Publication Type: Journal Article
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