5-Nitro-2,6-dioxohexahydro-4-pyrimidinecarboxamides: synthesis, in vitro antimycobacterial activity, cytotoxicity, and isocitrate lyase inhibition studies. [electronic resource]
Producer: 20110325Description: 765-72 p. digitalISSN:- 1475-6374
- Animals
- Anti-Bacterial Agents -- chemical synthesis
- Antitubercular Agents -- chemistry
- Bacterial Proteins -- antagonists & inhibitors
- Chlorocebus aethiops
- Computer Simulation
- Drug Evaluation, Preclinical
- Drug Resistance, Multiple, Bacterial
- Enzyme Inhibitors -- chemical synthesis
- Inhibitory Concentration 50
- Isocitrate Lyase -- antagonists & inhibitors
- Ligands
- Microbial Sensitivity Tests
- Molecular Structure
- Mycobacterium -- drug effects
- Mycobacterium smegmatis -- drug effects
- Mycobacterium tuberculosis -- drug effects
- Piperazines
- Protein Binding
- Pyrimidines -- chemical synthesis
- Quinolines
- Tuberculosis -- drug therapy
- Vero Cells
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
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