In vitro and in vivo characterization of A-940894: a potent histamine H4 receptor antagonist with anti-inflammatory properties. [electronic resource]
Producer: 20090617Description: 44-54 p. digitalISSN:- 1476-5381
- Animals
- Anti-Inflammatory Agents, Non-Steroidal -- pharmacokinetics
- Binding, Competitive
- Calcium -- metabolism
- Cell Shape
- Chemotaxis
- Eosinophils -- drug effects
- Female
- Histamine -- pharmacology
- Humans
- Male
- Mast Cells -- cytology
- Mice
- Mice, Inbred BALB C
- Peritonitis -- chemically induced
- Piperazines -- pharmacokinetics
- Prostaglandin D2 -- metabolism
- Pyrimidines -- pharmacokinetics
- RNA, Messenger -- biosynthesis
- Radioligand Assay
- Rats
- Rats, Sprague-Dawley
- Receptors, G-Protein-Coupled -- antagonists & inhibitors
- Receptors, Histamine -- biosynthesis
- Receptors, Histamine H4
- Recombinant Proteins -- antagonists & inhibitors
- Zymosan
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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