2-aryloxy-4-alkylaminopyridines: discovery of novel corticotropin-releasing factor 1 antagonists. [electronic resource]
Producer: 20080605Description: 1385-92 p. digitalISSN:- 0022-2623
- Action Potentials -- drug effects
- Administration, Oral
- Adrenocorticotropic Hormone -- blood
- Aminopyridines -- chemical synthesis
- Animals
- Antidepressive Agents -- chemical synthesis
- Cerebral Cortex -- metabolism
- Corticotropin-Releasing Hormone -- pharmacology
- Dogs
- Fasting
- Humans
- Injections, Intravenous
- Locus Coeruleus -- physiology
- Male
- Pituitary Gland -- metabolism
- Postprandial Period
- Radioligand Assay
- Rats
- Rats, Sprague-Dawley
- Receptors, Corticotropin-Releasing Hormone -- antagonists & inhibitors
- Reflex, Startle -- drug effects
- Structure-Activity Relationship
- CRF Receptor, Type 1
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Publication Type: Journal Article
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