ABP688, a novel selective and high affinity ligand for the labeling of mGlu5 receptors: identification, in vitro pharmacology, pharmacokinetic and biodistribution studies. [electronic resource]
Producer: 20070313Description: 903-14 p. digitalISSN:- 0968-0896
- Animals
- Autoradiography
- Binding, Competitive -- drug effects
- Blood Proteins -- metabolism
- Cell Line
- Chemical Phenomena
- Chemistry, Physical
- Cricetinae
- Excitatory Amino Acid Agonists -- pharmacology
- Humans
- In Vitro Techniques
- Indicators and Reagents
- Injections, Intravenous
- Ligands
- Male
- Mass Spectrometry
- Microsomes, Liver -- drug effects
- Oximes -- pharmacokinetics
- Phosphatidylinositols -- metabolism
- Positron-Emission Tomography
- Protein Binding
- Pyridines -- pharmacokinetics
- Quisqualic Acid -- antagonists & inhibitors
- Radiopharmaceuticals -- chemical synthesis
- Rats
- Rats, Sprague-Dawley
- Rats, Wistar
- Receptors, Kainic Acid -- drug effects
- Tissue Distribution
No physical items for this record
Publication Type: Journal Article
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