Synthesis and biological evaluation of the binding of dopamine D2/D3 receptor agonist, (R,S)-5-hydroxy-2-(N-propyl-N-(5'-(18)F-fluoropentyl)aminotetralin ((18)F-5-OH-FPPAT) in rodents and nonhuman primates. [electronic resource]
Producer: 20041221Description: 303-11 p. digitalISSN:- 0969-8051
- Animals
- Brain -- diagnostic imaging
- Dopamine D2 Receptor Antagonists
- Drug Evaluation, Preclinical
- Humans
- Isotope Labeling -- methods
- Kinetics
- Macaca mulatta
- Male
- Metabolic Clearance Rate
- Positron-Emission Tomography -- methods
- Primates
- Protein Binding
- Radiopharmaceuticals -- chemical synthesis
- Rats
- Rats, Sprague-Dawley
- Receptors, Dopamine D2 -- metabolism
- Receptors, Dopamine D3
- Rodentia
- Species Specificity
- Tetrahydronaphthalenes -- chemistry
- Tissue Distribution
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Publication Type: Comparative Study; Evaluation Study; Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
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