A cocaine insensitive chimeric insect serotonin transporter reveals domains critical for cocaine interaction. [electronic resource]
Producer: 20021010Description: 3934-44 p. digitalISSN:- 0014-2956
- Amino Acid Sequence
- Animals
- Biological Transport -- drug effects
- Carrier Proteins -- antagonists & inhibitors
- Cell Line
- Chlorides -- pharmacology
- Chlorocebus aethiops
- Cloning, Molecular
- Cocaine -- pharmacology
- Drug Resistance
- Fluoxetine -- pharmacology
- Humans
- Hydrophobic and Hydrophilic Interactions
- Insect Proteins -- antagonists & inhibitors
- Manduca -- chemistry
- Membrane Glycoproteins -- antagonists & inhibitors
- Membrane Transport Proteins
- Molecular Sequence Data
- Mutagenesis, Site-Directed
- Nerve Tissue Proteins -- antagonists & inhibitors
- Protein Conformation
- Protein Structure, Tertiary
- Recombinant Fusion Proteins -- antagonists & inhibitors
- Sequence Alignment
- Sequence Homology, Amino Acid
- Serotonin -- metabolism
- Serotonin Antagonists -- metabolism
- Serotonin Plasma Membrane Transport Proteins
- Serotonin Receptor Agonists -- metabolism
- Selective Serotonin Reuptake Inhibitors -- pharmacology
- Sodium -- pharmacology
- Species Specificity
- Structure-Activity Relationship
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Publication Type: Comparative Study; Journal Article; Research Support, U.S. Gov't, P.H.S.
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